Synthesis and Elastase Inhibitory Evaluation of Phosphate Esters and Mixed Phosphate Anhydride of Penam Sulfones

Abstract

The evaluation of human leucocite elastase inhibition by phosphate esters (1-2) and phosphate mixed anhydride (3) of penicillin sulfones and their precursor sulfides is described.

Keywords

• Elastase Inhibition
• Phosphate Esters
• Phosphate Anhydride
• Penam Sulfones