An Improved Synthetic Process of Two Key Intermediates and Their Application in the Synthesis of Lifitegrast

• Gang-Long Jiang,
• Xin-Kun Wang,
• Xiao-Fei Xiao,
• Yu Liu

Affiliations

Gang-Long Jiang

Incubation Centre of S&T Achievements, Shanghai Institute of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai, People's Republic of China

Xin-Kun Wang

College of Chemistry and Chemical Engineering, Shanghai University of Engineering Science, Shanghai, People's Republic of China

Xiao-Fei Xiao

Incubation Centre of S&T Achievements, Shanghai Institute of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai, People's Republic of China

Yu Liu

Incubation Centre of S&T Achievements, Shanghai Institute of Pharmaceutical Industry, China State Institute of Pharmaceutical Industry Co., Ltd., Shanghai, People's Republic of China