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CHIMIA
(Mar 2022)
Late-stage Functionalization and its Impact on Modern Drug Discovery
David F. Nippa,
Remo Hohler,
Antonia F. Stepan,
Uwe Grether,
David B. Konrad,
Rainer E. Martin
Affiliations
David F. Nippa
Department of Pharmacy, Ludwigs-Maximilians-Universität München; F. Hoffmann-La Roche Ltd., Basel
Remo Hohler
Department of Pharmacy, Ludwigs-Maximilians-Universität München; F. Hoffmann-La Roche Ltd., Basel
Antonia F. Stepan
F. Hoffmann-La Roche Ltd., Basel
Uwe Grether
F. Hoffmann-La Roche Ltd., Basel
David B. Konrad
Department of Pharmacy, Ludwigs-Maximilians-Universität München
Rainer E. Martin
F. Hoffmann-La Roche Ltd., Basel
DOI
https://doi.org/10.2533/chimia.2022.258
Journal volume & issue
Vol. 76, no. 3
Abstract
Read online
No abstracts available.
Keywords
Catalysis
Diversification
Late-stage functionalization
Medicinal chemistry
Synthesis
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