Enantioselective Synthesis of (R)‑Sitagliptin via Phase-Transfer Catalytic aza-Michael Addition

• Daehyun Oh,
• Jaeyong Lee,
• Sehun Yang,
• So Hyun Jung,
• Mihyun Kim,
• Geumwoo Lee,
• Hyeung-geun Park

Affiliations

Daehyun Oh

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea

Jaeyong Lee

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea

Sehun Yang

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea

So Hyun Jung

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea

Mihyun Kim

College of Pharmacy, Gachon University, Incheon, Republic of Korea

Geumwoo Lee

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea

Hyeung-geun Park

Research Institute of Pharmaceutical Sciences and College of Pharmacy, Seoul National University, Seoul, Republic of Korea