Progress Toward a Large-Scale Synthesis of Molnupiravir (MK-4482, EIDD-2801) from Cytidine

• Grace P. Ahlqvist,
• Catherine P. McGeough,
• Chris Senanayake,
• Joseph D. Armstrong,
• Ajay Yadaw,
• Sarabindu Roy,
• Saeed Ahmad,
• David R. Snead,
• Timothy F. Jamison

Affiliations

Grace P. Ahlqvist

Department of Chemistry, Massachusetts Institute of Technology, Cambridge, Massachusetts, United States

Catherine P. McGeough

Department of Chemistry, Massachusetts Institute of Technology, Cambridge, Massachusetts, United States

Chris Senanayake

TCG GreenChem, Inc., Process R&D Center at Princeton South, Ewing, New Jersey, United States

Joseph D. Armstrong

TCG GreenChem, Inc., Process R&D Center at Princeton South, Ewing, New Jersey, United States

Ajay Yadaw

TCG GreenChem, Inc., Process R&D Center at Princeton South, Ewing, New Jersey, United States

Sarabindu Roy

TCG GreenChem, Inc., Process R&D Center at Princeton South, Ewing, New Jersey, United States

Saeed Ahmad

Medicines for All Institute, Richmond, Virginia, United States

David R. Snead

Medicines for All Institute, Richmond, Virginia, United States

Timothy F. Jamison

Department of Chemistry, Massachusetts Institute of Technology, Cambridge, Massachusetts, United States